{"id":9950,"date":"2025-09-26T16:20:22","date_gmt":"2025-09-26T14:20:22","guid":{"rendered":"https:\/\/rvh-synergie.org\/actualites\/la-science-ouverte-donne-un-coronavirus-a-large-spectre-antiviral\/"},"modified":"2025-09-26T16:20:25","modified_gmt":"2025-09-26T14:20:25","slug":"la-science-ouverte-donne-un-coronavirus-a-large-spectre-antiviral","status":"publish","type":"post","link":"https:\/\/rvh-synergie.org\/actualites\/la-science-ouverte-donne-un-coronavirus-a-large-spectre-antiviral\/","title":{"rendered":"La science ouverte donne un coronavirus \u00e0 large spectre antiviral"},"content":{"rendered":"<div>\n<div class=\"article-gallery lightGallery\">\n<div data-thumb=\"https:\/\/scx1.b-cdn.net\/csz\/news\/tmb\/2022\/microscope-4.jpg\" data-src=\"https:\/\/scx2.b-cdn.net\/gfx\/news\/hires\/2022\/microscope-4.jpg\" data-sub-html=\"Credit: Pixabay\/CC0 Public Domain\">\n<figure class=\"article-img\">\n<\/figure><\/div>\n<\/div>\n<p>Un nouvel coronavirus \u00e0 large spectre antiviral, ASAP-0017445, a \u00e9t\u00e9 nomm\u00e9 candidat pr\u00e9clinique sur le m\u00e9dicament par les m\u00e9dicaments pour les maladies n\u00e9glig\u00e9es (DNDI).<\/p>\n<p>Le candidat est le premier coronavirus antiviral d\u00e9velopp\u00e9 par le crowdsourcing et la science ouverte, et le premier avec ses origines dans l&rsquo;intelligence artificielle (IA). Le candidat est le r\u00e9sultat d&rsquo;une recherche de l&rsquo;initiative Covid Moonshot qui est originaire de Diamond Light Source.<\/p>\n<p>Il s&rsquo;agit d&rsquo;un principal inhibiteur de la prot\u00e9ase qui montre une activit\u00e9 prometteuse contre le SRAS-COV2 et d&rsquo;autres virus de la m\u00eame famille, y compris d&rsquo;autres virus de potentiel pand\u00e9mique tels que Merscov &#8211; d&rsquo;o\u00f9 sa qualification de spectre \u00e0 large. Le compos\u00e9 a \u00e9t\u00e9 con\u00e7u et d\u00e9velopp\u00e9 par Covid Moonshot Covid Moonshot et son organisation s\u0153ur, le consortium antiviral (ASAP), le consortium AI-A-ax\u00e9 sur la structure AI.<\/p>\n<p>\u00ab\u00a0Notre objectif est de fournir une m\u00e9decine antivirale efficace et abordable qui serait accessible \u00e0 tout le monde si et quand la prochaine pand\u00e9mie de coronavirus frappe\u00a0\u00bb, a d\u00e9clar\u00e9 Annette von Delft, chef des anti-infectices au centre de la d\u00e9couverte des m\u00e9dicaments, \u00e0 l&rsquo;Universit\u00e9 d&rsquo;Oxford et partenaire de l&rsquo;initiative Moonshot.<\/p>\n<p>Le Moonshot covide \u00e9tait une collaboration mondiale spontan\u00e9e qui a commenc\u00e9 en mars 2020, d\u00e9clench\u00e9 par les donn\u00e9es de la plate-forme Xchem de Diamond pour le d\u00e9pistage des fragments. Des chercheurs du monde entier ont soumis plus de 18 000 conceptions de mol\u00e9cules pour inhiber la principale prot\u00e9ase du SARS-COV-2.<\/p>\n<p>Les structures d\u00e9taill\u00e9es ont \u00e9t\u00e9 mises \u00e0 disposition ouvertement, garantissant que chaque \u00e9tape du processus de d\u00e9couverte pourrait \u00eatre construite par la communaut\u00e9 de la recherche mondiale. Cet engagement envers la transparence et les donn\u00e9es ouvertes a jet\u00e9 les bases de l&rsquo;optimisation d&rsquo;ASAP-0017445.<\/p>\n<p>La contribution de Diamond souligne l&rsquo;importance de l&rsquo;infrastructure de recherche avanc\u00e9e dans l&rsquo;acc\u00e9l\u00e9ration de la d\u00e9couverte de m\u00e9dicaments. En combinant la cristallographie, la mod\u00e9lisation informatique et la conception mondiale de crowdsourced, le Moonshot a d\u00e9montr\u00e9 comment la collaboration ouverte peut livrer un candidat de m\u00e9dicament destin\u00e9 \u00e0 \u00eatre directement \u00e0 la g\u00e9n\u00e9ration et \u00e0 mondialement accessible.<\/p>\n<p>La structure d&rsquo;ASAP-0017445 a \u00e9t\u00e9 divulgu\u00e9e publiquement en mars 2025. Toutes les donn\u00e9es g\u00e9n\u00e9r\u00e9es au cours de son d\u00e9veloppement, y compris les donn\u00e9es de structure des plus de 2 000 compos\u00e9s soumises pendant la phase de crowdsourcing, sont accessibles au public. D&rsquo;autres chercheurs peuvent s&rsquo;appuyer sur cet ensemble de donn\u00e9es sans pr\u00e9c\u00e9dent pour la d\u00e9couverte de m\u00e9dicaments pour leurs propres recherches.<\/p>\n<p>                                        <!-- print only --><\/p><\/div>\n","protected":false},"excerpt":{"rendered":"<p>Un nouvel coronavirus \u00e0 large spectre antiviral, ASAP-0017445, a \u00e9t\u00e9 nomm\u00e9 candidat pr\u00e9clinique sur le<\/p>\n","protected":false},"author":1,"featured_media":9951,"comment_status":"closed","ping_status":"","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[86],"tags":[3601,4451,2633,3418,6810,2022,786],"class_list":["post-9950","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-les-maladies","tag-antiviral","tag-coronavirus","tag-donne","tag-large","tag-ouverte","tag-science","tag-spectre","generate-columns","tablet-grid-50","mobile-grid-100","grid-parent","grid-50","resize-featured-image"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.4 - 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