{"id":8967,"date":"2025-08-28T23:58:47","date_gmt":"2025-08-28T21:58:47","guid":{"rendered":"https:\/\/rvh-synergie.org\/actualites\/explorer-la-promesse-des-cellules-ipsc-humaines-pour-comprendre-les-abus-de-fentanyl\/"},"modified":"2025-08-28T23:58:48","modified_gmt":"2025-08-28T21:58:48","slug":"explorer-la-promesse-des-cellules-ipsc-humaines-pour-comprendre-les-abus-de-fentanyl","status":"publish","type":"post","link":"https:\/\/rvh-synergie.org\/actualites\/explorer-la-promesse-des-cellules-ipsc-humaines-pour-comprendre-les-abus-de-fentanyl\/","title":{"rendered":"Explorer la promesse des cellules IPSC humaines pour comprendre les abus de fentanyl"},"content":{"rendered":"<div>\n<div class=\"article-gallery lightGallery\">\n<div data-thumb=\"https:\/\/scx1.b-cdn.net\/csz\/news\/tmb\/2025\/exploring-the-promise.jpg\" data-src=\"https:\/\/scx2.b-cdn.net\/gfx\/news\/2025\/exploring-the-promise.jpg\" data-sub-html=\"Credit: &lt;i&gt;Circulation&lt;\/i&gt; (2025). DOI: 10.1161\/CIRCULATIONAHA.123.068560\">\n<figure class=\"article-img\">\n<\/figure><\/div>\n<\/div>\n<p>Ces derni\u00e8res ann\u00e9es, le fentanyl, un opio\u00efde synth\u00e9tique de 50 \u00e0 100 fois plus fort que la morphine, a \u00e9t\u00e9 un contributeur principal \u00e0 la crise des opio\u00efdes. L&rsquo;un des pires effets n\u00e9fastes de l&rsquo;abus de fentanyl est l&rsquo;arr\u00eat cardiaque induit par les opio\u00efdes. Bien qu&rsquo;il soit bien connu que l&rsquo;abus d&rsquo;opio\u00efdes peut induire des arythmies, les effets de l&rsquo;abus de fentanyl sur les rythmes cardiaques n&rsquo;ont pas encore \u00e9t\u00e9 enti\u00e8rement \u00e9tudi\u00e9s.<\/p>\n<p>Dans une \u00e9tude r\u00e9cente publi\u00e9e dans <i>Circulation<\/i>premier auteur Gema Mond\u00e9jar-Parre\u00f1o, Ph.D. et l&rsquo;auteur principal Joseph C. Wu, MD, Ph.D., directeur du Stanford Cardiovascular Institute, a constat\u00e9 que les cellules souches pluripotentes induites par l&rsquo;homme offrent une occasion in\u00e9gal\u00e9e d&rsquo;\u00e9tudier les r\u00e9ponses sp\u00e9cifiques au patient \u00e0 l&rsquo;abus d&rsquo;opio\u00efdes.<\/p>\n<p>Les enqu\u00eateurs ont \u00e9tudi\u00e9 les cons\u00e9quences de la maltraitance du fentanyl, en particulier celles li\u00e9es \u00e0 l&rsquo;activit\u00e9 \u00e9lectrique du c\u0153ur, qui d\u00e9terminent comment le c\u0153ur contr\u00f4le son rythme et son pompage. Les scientifiques ont analys\u00e9 19 \u00e9tudes de toxicologie entre 1994 et 2022 dans lesquelles l&rsquo;estimation moyenne de la concentration de fentanyl \u00e9tait trois fois plus \u00e9lev\u00e9e que pour les patients souffrant de douleur chronique. En utilisant les donn\u00e9es, les chercheurs ont expos\u00e9 des cardiomyocytes d\u00e9riv\u00e9s des cellules souches induits par l&rsquo;homme (IPSC-CM) \u00e0 des doses de fentanyl qui imitaient les circonstances de surdose.<\/p>\n<p>Ils ont constat\u00e9 que cela provoquait des changements dans la signalisation du calcium de l&rsquo;hom\u00e9ostasie dans les cellules musculaires cardiaques et a ralenti la pr\u00e9paration du rythme cardiaque suivant, ce qui a contribu\u00e9 \u00e0 battre les irr\u00e9gularit\u00e9s. De plus, comme les arythmies sont souvent plus \u00e9videntes lorsque la fr\u00e9quence cardiaque augmente, les chercheurs ont trouv\u00e9 la combinaison du fentanyl et de l&rsquo;isoprot\u00e9r\u00e9nol, un stimulant utilis\u00e9 pour augmenter la fr\u00e9quence cardiaque, peut aggraver les arythmies induites par le fentanyl.<\/p>\n<p>Cette \u00e9tude fournit des preuves que les abus de fentanyl peuvent alt\u00e9rer la fonction des cellules cardiaques, conduisant \u00e0 des d\u00e9fauts de rythme. Avec la d\u00e9pression respiratoire, les effets induits par le fentanyl sur l&rsquo;\u00e9lectrophysiologie contribuent consid\u00e9rablement \u00e0 un arr\u00eat cardiaque. D&rsquo;autres \u00e9tudes nous aideront \u00e0 mieux comprendre les abus de fentanyl et sa relation avec les arythmies.<\/p>\n<p>                                        <!-- print only --><\/p><\/div>\n","protected":false},"excerpt":{"rendered":"<p>Ces derni\u00e8res ann\u00e9es, le fentanyl, un opio\u00efde synth\u00e9tique de 50 \u00e0 100 fois plus fort<\/p>\n","protected":false},"author":1,"featured_media":8968,"comment_status":"closed","ping_status":"","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[35],"tags":[4605,1622,310,16,1502,328,227,6023,49,8,4708],"class_list":["post-8967","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-les-addictions","tag-abus","tag-cellules","tag-comprendre","tag-des","tag-explorer","tag-fentanyl","tag-humaines","tag-ipsc","tag-les","tag-pour","tag-promesse","generate-columns","tablet-grid-50","mobile-grid-100","grid-parent","grid-50","resize-featured-image"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.4 - 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