{"id":7073,"date":"2025-06-05T23:56:21","date_gmt":"2025-06-05T21:56:21","guid":{"rendered":"https:\/\/rvh-synergie.org\/actualites\/une-nouvelle-approche-inverse-les-surdoses-opioides-plus-en-toute-securite-montre-letude-de-rat\/"},"modified":"2025-06-05T23:56:23","modified_gmt":"2025-06-05T21:56:23","slug":"une-nouvelle-approche-inverse-les-surdoses-opioides-plus-en-toute-securite-montre-letude-de-rat","status":"publish","type":"post","link":"https:\/\/rvh-synergie.org\/actualites\/une-nouvelle-approche-inverse-les-surdoses-opioides-plus-en-toute-securite-montre-letude-de-rat\/","title":{"rendered":"Une nouvelle approche inverse les surdoses opio\u00efdes plus en toute s\u00e9curit\u00e9, montre l&rsquo;\u00e9tude de rat"},"content":{"rendered":"<div>\n<div class=\"article-gallery lightGallery\">\n<div data-thumb=\"https:\/\/scx1.b-cdn.net\/csz\/news\/tmb\/2025\/new-approach-reverses.jpg\" data-src=\"https:\/\/scx2.b-cdn.net\/gfx\/news\/2025\/new-approach-reverses.jpg\" data-sub-html=\"Blocking opioid receptors outside the brain reverses opioid overdose without sudden and severe withdrawal symptoms. Credit: &lt;i&gt;eLife&lt;\/i&gt; (2025). DOI: 10.7554\/eLife.104469.3\">\n<figure class=\"article-img\">\n<\/figure><\/div>\n<\/div>\n<p>Les surdoses d&rsquo;opio\u00efdes sont un probl\u00e8me majeur de sant\u00e9 publique aux \u00c9tats-Unis, tuant des dizaines de milliers de personnes chaque ann\u00e9e. Le m\u00e9dicament naloxone, qui est disponible en tant que spray nasal en vente libre ou donn\u00e9 par injection, a sauv\u00e9 d&rsquo;innombrables vies en inversant rapidement les surdoses d&rsquo;opio\u00efdes. Mais pour bloquer les r\u00e9cepteurs opio\u00efdes dans le cerveau, la naloxone provoque de graves sympt\u00f4mes de sevrage, notamment la douleur, les vomissements et l&rsquo;agitation.<\/p>\n<p>Une \u00e9quipe de recherche du laboratoire deoipcion de cr\u00e9tin de Washu Medicine a d\u00e9couvert une nouvelle fa\u00e7on prometteuse de traiter les surdoses d&rsquo;opio\u00efdes sans d\u00e9clencher de sympt\u00f4mes de sevrage graves. Leur \u00e9tude, intitul\u00e9e \u00ab\u00a0L&rsquo;antagonisme des r\u00e9cepteurs opio\u00efdes p\u00e9riph\u00e9riques att\u00e9nue la d\u00e9pression cardiorespiratoire induite par le fentanyl et est d\u00e9pourvue de comportement aversif\u00a0\u00bb, est publi\u00e9 dans <i>elife<\/i>.<\/p>\n<p>Le travail montre que le ciblage des r\u00e9cepteurs opio\u00efdes \u00e0 l&rsquo;ext\u00e9rieur du cerveau peut inverser efficacement les effets de surdosage sans provoquer l&rsquo;inconfort intense typique des traitements actuels.<\/p>\n<p>Dirig\u00e9e par Jose Moron-Concepcion, Ph.D., et Brian Ruyle, Ph.D., les chercheurs ont test\u00e9 un m\u00e9dicament appel\u00e9 Naloxone-Methiodure, qui est similaire \u00e0 la naloxone mais ne traverse pas la barri\u00e8re h\u00e9mato-enc\u00e9phalique et se concentre plut\u00f4t sur le corps. Dans l&rsquo;\u00e9tude, ils ont constat\u00e9 que la naloxone-m\u00e9thodiodide pouvait inverser efficacement la d\u00e9pression respiratoire induite par le fentanyl sans d\u00e9clencher les sympt\u00f4mes de sevrage graves associ\u00e9s \u00e0 la naloxone.<\/p>\n<p>\u00ab\u00a0Ces r\u00e9sultats ont un impact potentiel important \u00e9tant donn\u00e9 que le fentanyl est toujours le principal moteur des d\u00e9c\u00e8s li\u00e9s aux opio\u00efdes dans ce pays\u00a0\u00bb, a d\u00e9clar\u00e9 Moron-Concepcion. \u00ab\u00a0Notre nouvelle approche th\u00e9rapeutique est prometteuse en r\u00e9duisant les effets ind\u00e9sirables g\u00e9n\u00e9ralement observ\u00e9s avec la naloxone, offrant un moyen plus s\u00fbr d&rsquo;inverser les surdoses.\u00a0\u00bb<\/p>\n<p>Cette d\u00e9couverte ouvre la possibilit\u00e9 de traitements de surdose plus s\u00fbrs et plus humains, contribuant \u00e0 r\u00e9duire la peur et la stigmatisation qui emp\u00eachent souvent les gens de rechercher des soins de sauvetage.<\/p>\n<p>                                        <!-- print only --><\/p><\/div>\n","protected":false},"excerpt":{"rendered":"<p>Les surdoses d&rsquo;opio\u00efdes sont un probl\u00e8me majeur de sant\u00e9 publique aux \u00c9tats-Unis, tuant des dizaines<\/p>\n","protected":false},"author":1,"featured_media":7074,"comment_status":"closed","ping_status":"","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[35],"tags":[1426,4125,49,1346,210,244,411,1059,448,291,137,47],"class_list":["post-7073","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-les-addictions","tag-approche","tag-inverse","tag-les","tag-letude","tag-montre","tag-nouvelle","tag-opioides","tag-rat","tag-securite","tag-surdoses","tag-toute","tag-une","generate-columns","tablet-grid-50","mobile-grid-100","grid-parent","grid-50","resize-featured-image"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.4 - 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