{"id":1943,"date":"2024-11-07T02:49:52","date_gmt":"2024-11-07T01:49:52","guid":{"rendered":"https:\/\/rvh-synergie.org\/actualites\/la-decouverte-du-mecanisme-de-replication-rapide-du-covid-19-pourrait-elargir-les-options-de-traitement\/"},"modified":"2024-11-07T02:49:54","modified_gmt":"2024-11-07T01:49:54","slug":"la-decouverte-du-mecanisme-de-replication-rapide-du-covid-19-pourrait-elargir-les-options-de-traitement","status":"publish","type":"post","link":"https:\/\/rvh-synergie.org\/actualites\/la-decouverte-du-mecanisme-de-replication-rapide-du-covid-19-pourrait-elargir-les-options-de-traitement\/","title":{"rendered":"La d\u00e9couverte du m\u00e9canisme de r\u00e9plication rapide du COVID-19 pourrait \u00e9largir les options de traitement"},"content":{"rendered":"<div>\n<div class=\"article-gallery lightGallery\">\n<div data-thumb=\"https:\/\/scx1.b-cdn.net\/csz\/news\/tmb\/2024\/discovery-of-rapid-cov.jpg\" data-src=\"https:\/\/scx2.b-cdn.net\/gfx\/news\/hires\/2024\/discovery-of-rapid-cov.jpg\" data-sub-html=\"A schematic diagram showing the significant contribution of SCoV2-induced altered mitochondrial dynamics and mitochondrial EGFR translocation in sustaining viral propagation. First, SCoV2 RNA and nucleocapsid complex increases membrane potential during the early stages of SCoV2 infection. This alteration subsequently promotes mitochondrial elongation. SCoV2 also activates the mitochondrial OXPHOS process, thereby promoting ATP production. Second, SCoV2 activates EGFR-mediated cell survival signaling and subsequently promotes mitochondrial EGFR internalization, which contributes to the maintenance of abnormal mitochondrial bioenergetics. These alterations are physiologically relevant to the maintenance of homoeostasis of SCoV2-infected cells and robust SCoV2 propagation. Credit: Korea Research Institute of Chemical Technology (KRICT)\">\n<figure class=\"article-img\">\n<\/figure><\/div>\n<\/div>\n<p>Les inqui\u00e9tudes concernant le COVID-19 ont consid\u00e9rablement diminu\u00e9, mais les chercheurs continuent d\u2019analyser son taux de transmission \u00e9lev\u00e9, dans le but de se pr\u00e9parer \u00e0 de futures maladies infectieuses. Une \u00e9quipe de recherche a r\u00e9cemment identifi\u00e9 le m\u00e9canisme \u00e0 l\u2019origine de la prolif\u00e9ration rapide du virus COVID-19.<\/p>\n<p>L&rsquo;\u00e9quipe du Dr Seong-Jun Kim de l&rsquo;Institut cor\u00e9en de recherche en technologie chimique (KRICT) a rapport\u00e9 dans un document de recherche que la prolif\u00e9ration rapide du COVID-19 est due \u00e0 une modification des r\u00f4les des mitochondries et du r\u00e9cepteur du facteur de croissance \u00e9pidermique (EGFR ; responsable de la croissance). transmission du signal dans les cellules).<\/p>\n<p>L&rsquo;article est publi\u00e9 dans la revue <i>Transduction du signal et th\u00e9rapie cibl\u00e9e<\/i>.<\/p>\n<p>Des coronavirus \u00e0 l\u2019origine de pand\u00e9mies, tels que le SRAS en 2003, le MERS en 2015 et le COVID-19 en 2019, sont apparus \u00e0 plusieurs reprises. Compte tenu de la fr\u00e9quence croissante de ces \u00e9pid\u00e9mies, il est urgent d\u2019acc\u00e9l\u00e9rer la r\u00e9ponse aux nouvelles maladies infectieuses.<\/p>\n<p>Alors que de nombreuses \u00e9tudes sur le COVID-19 ont \u00e9t\u00e9 men\u00e9es, se concentrant initialement sur le m\u00e9canisme d\u2019entr\u00e9e du virus et le d\u00e9veloppement de vaccins, des recherches r\u00e9centes ont explor\u00e9 des m\u00e9thodes permettant d\u2019entraver la r\u00e9plication virale en modifiant les concentrations d\u2019ions calcium dans les cellules.<\/p>\n<p>Cependant, le m\u00e9canisme pr\u00e9cis qui sous-tend la r\u00e9plication rapide du virus apr\u00e8s son entr\u00e9e dans les cellules humaines reste flou. Comprendre ce processus est crucial pour la pr\u00e9paration \u00e0 une future pand\u00e9mie.<\/p>\n<p>L&rsquo;\u00e9quipe du Dr Kim a r\u00e9v\u00e9l\u00e9 qu&rsquo;une fois que le COVID-19 envahit les cellules humaines, il modifie rapidement la structure et la fonction des mitochondries pour augmenter anormalement la production d&rsquo;\u00e9nergie, essentielle \u00e0 la r\u00e9plication virale. Ils ont \u00e9galement d\u00e9couvert que le virus manipule la prot\u00e9ine EGFR, essentielle \u00e0 la signalisation de la croissance cellulaire, pour maintenir cette r\u00e9plication rapide.<\/p>\n<p>Cela augmente la probabilit\u00e9 que le virus se r\u00e9plique et se propage en grand nombre. Surtout, l\u2019\u00e9quipe a d\u00e9montr\u00e9 par des exp\u00e9riences que l\u2019utilisation de m\u00e9dicaments ciblant l\u2019EGFR pourrait traiter efficacement le COVID-19.<\/p>\n<div class=\"article-gallery lightGallery\">\n<div data-thumb=\"https:\/\/scx1.b-cdn.net\/csz\/news\/tmb\/2024\/discovery-of-rapid-cov-1.jpg\" data-src=\"https:\/\/scx2.b-cdn.net\/gfx\/news\/hires\/2024\/discovery-of-rapid-cov-1.jpg\" data-sub-html=\"\u25b2Lung tissue qRT-PCR test results three days after administration \u2192 Viral RNA reduced approximately 10-fold. The results of a staining test on the lung tissue inflammation area six days after administration, \u2192 Significantly alleviates lung inflammation. Credit: Korea Research Institute of Chemical Technology (KRICT)\">\n<figure class=\"article-img text-center\">\n            <img decoding=\"async\" src=\"https:\/\/rvh-synergie.org\/actualites\/wp-content\/uploads\/2024\/11\/1730944192_812_La-decouverte-du-mecanisme-de-replication-rapide-du-COVID-19-pourrait.jpg\" alt=\"D\u00e9couverte d\u2019un m\u00e9canisme de r\u00e9plication rapide du COVID-19 et d\u2019options de traitement \u00e9largies\" title=\"\u25b2R\u00e9sultats du test qRT-PCR du tissu pulmonaire trois jours apr\u00e8s l'administration \u2192 L'ARN viral est r\u00e9duit d'environ 10 fois. Les r\u00e9sultats d'un test de coloration sur la zone d'inflammation du tissu pulmonaire six jours apr\u00e8s l'administration, \u2192 Att\u00e9nue consid\u00e9rablement l'inflammation pulmonaire. Cr\u00e9dit\u00a0: Institut cor\u00e9en de recherche en technologie chimique (KRICT)\"><br \/>\n                     <\/figure>\n<\/p><\/div>\n<\/div>\n<p>Les chercheurs se sont concentr\u00e9s sur deux ph\u00e9nom\u00e8nes majeurs se produisant apr\u00e8s l\u2019entr\u00e9e du virus dans les cellules h\u00f4tes :<\/p>\n<ul>\n<li>Production am\u00e9lior\u00e9e d\u2019ATP\u00a0: le complexe viral ARN-nucl\u00e9ocapside influence le potentiel de la membrane mitochondriale, entra\u00eenant une augmentation anormale de la production d\u2019\u00e9nergie. La fusion des mitochondries est favoris\u00e9e, augmentant ainsi la surface et l\u2019efficacit\u00e9 de la production d\u2019ATP.<\/li>\n<li>Alt\u00e9ration de la fonction de l&rsquo;EGFR\u00a0: l&rsquo;infection au COVID-19 active la voie de signalisation de l&rsquo;EGFR, l&rsquo;EGFR modifi\u00e9 se d\u00e9pla\u00e7ant vers les mitochondries. Cela entretient une production d\u2019\u00e9nergie excessive, facilitant une r\u00e9plication virale rapide.<\/li>\n<\/ul>\n<p>En utilisant des inhibiteurs de l&rsquo;EGFR approuv\u00e9s par la FDA, tels que le vand\u00e9tanib et le dacomitinib, l&rsquo;\u00e9quipe a confirm\u00e9 des effets antiviraux significatifs. Le vand\u00e9tanib s\u2019est notamment r\u00e9v\u00e9l\u00e9 tr\u00e8s efficace, r\u00e9duisant de 90 % les niveaux d\u2019ARN viral chez les souris infect\u00e9es apr\u00e8s une administration orale pendant trois jours et att\u00e9nuant consid\u00e9rablement l\u2019inflammation pulmonaire apr\u00e8s six jours.<\/p>\n<p>De plus, l\u2019efficacit\u00e9 antivirale du vand\u00e9tanib contre les variantes du COVID-19 telles que alpha, b\u00eata, delta et omicron \u00e9tait remarquable, avec une r\u00e9duction jusqu\u2019\u00e0 100\u00a0000 fois des niveaux d\u2019ARN viral dans certains cas. Le vand\u00e9tanib a \u00e9galement emp\u00each\u00e9 efficacement l\u2019infection de la descendance virale nouvellement produite.<\/p>\n<p>Les r\u00e9sultats d\u00e9montrent un nouveau m\u00e9canisme sous-jacent \u00e0 la r\u00e9plication rapide du COVID-19 et sugg\u00e8rent le potentiel de r\u00e9utilisation des m\u00e9dicaments pour traiter les infections virales \u00e0 l&rsquo;aide de th\u00e9rapies approuv\u00e9es existantes. Cette d\u00e9couverte pourrait constituer une \u00e9tape importante dans la lutte contre les futures maladies infectieuses.<\/p>\n<p>Le Dr Kim du KRICT a d\u00e9clar\u00e9 : \u00ab \u00c0 l&rsquo;heure o\u00f9 nous devons nous pr\u00e9parer \u00e0 la propagation fr\u00e9quente des maladies infectieuses, l&rsquo;identification d&rsquo;un nouveau m\u00e9canisme de r\u00e9plication virale rapide et le d\u00e9veloppement de nouvelles strat\u00e9gies de traitement contribueront \u00e0 la sant\u00e9 et \u00e0 la s\u00e9curit\u00e9 des personnes. personnes.\u00a0\u00bb<\/p>\n<p>                                        <!-- print only --><\/p><\/div>\n","protected":false},"excerpt":{"rendered":"<p>Les inqui\u00e9tudes concernant le COVID-19 ont consid\u00e9rablement diminu\u00e9, mais les chercheurs continuent d\u2019analyser son taux<\/p>\n","protected":false},"author":1,"featured_media":1944,"comment_status":"closed","ping_status":"","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[86],"tags":[561,2305,2307,49,1256,950,203,1533,2306,261],"class_list":["post-1943","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-les-maladies","tag-covid19","tag-decouverte","tag-elargir","tag-les","tag-mecanisme","tag-options","tag-pourrait","tag-rapide","tag-replication","tag-traitement","generate-columns","tablet-grid-50","mobile-grid-100","grid-parent","grid-50","resize-featured-image"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.4 - 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Depuis plus de dix ans, j'explore et rapporte les histoires poignantes des individus confront\u00e9s \u00e0 ces d\u00e9fis, tout en sensibilisant le public aux traitements novateurs et aux progr\u00e8s scientifiques dans ce domaine. 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